Home Tools
Log in
Cart

Search Result

Search Results for " estrogen receptor modulator 1 "

8

Compounds

Cat No. Product Name Synonyms Targets
T15249 Estrogen receptor modulator 1 Estrogen Receptor/ERR
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.4...
T2569 Chlorotrianisene tris(p-methoxyphenyl)chloroethylene,CTA,tri-p-anisylchloroethylene,TACE Estrogen Receptor/ERR , Estrogen/progestogen Receptor , COX
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen receptor modulator (SERM), with predominantly estrogenic but...
T79064 Estrogen receptor modulator 7 Estrogen Receptor/ERR
Estrogen Receptor Modulator 7 is a potent modulator of estrogen receptors, utilized in cancer research [1].
T25700 Levormeloxifene
Levormeloxifene is a selective modulator of the estrogen receptor. It inhibits the production of vaginal tropoelastin and transforming growth factor-beta 1.
T79109 Estrogen receptor modulator 8 Estrogen Receptor/ERR
Estrogen Receptor Modulator 8 (compound 4) is an orally active inhibitor targeting Estrogen Receptor/ERR α with potent efficacy (IC50 = 0.437 nM in MCF-7 cells) and effectively hampers MCF-7 cell proliferation (IC50 = 0....
T60674 DK1
DK1 is a potent estrogen related receptor modulator. DK1 impacts the activity of ERRα receptor and reduces blood glucose. DK1 shows the potential in the diabetes research [1].
T79382 ER degrader 6 Estrogen Receptor/ERR
ER degrader 6 (compound 35s) is a potent selective estrogen receptor modulator (SERM) with the capacity to degrade Estrogen Receptor (ER)α. It disrupts the microtubule network, inhibiting tubulin polymerization, and effe...
T82439 Estrogen receptor modulator 10 Estrogen Receptor/ERR
Compound G-5b, an estrogen receptor modulator 10, functions as an estrogen receptor (ER) antagonist (IC50=6.7 nM) and degrader (DC50=0.4 nM). It has the capability to induce apoptosis and block cells at the G1/G0 phase, ...
TargetMol